SCHEMBL20176823

SCHEMBL20176823

Cc1cn(-c2ccc(Br)cc2)ccc1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.46
HPGD P15428 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HSD17B10 Q99714 1/20 0.46
FAAH O00519 1/20 0.42
MGLL Q99685 1/20 0.42
COMT P21964 2/20 0.41
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
KAT2B Q92831 1/20 0.35
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.33
NLRP3 Q96P20 1/20 0.33
HCAR1 Q9BXC0 1/20 0.33
HSP90AA1 P07900 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14827196 0.81 COMT (0.61) HPGDHSD17B10MGLLCOMTGSK3A
SCHEMBL27617592 0.78 HPGD (0.47) POLBHPGDNPSR1HSD17B10FAAH
SCHEMBL21579385 0.74 FAAH (0.43) FAAHMGLLCOMT
SCHEMBL20176828 0.74 COMT (0.41) HPGDNPSR1HSD17B10FAAHMGLL
SCHEMBL20176822 0.74 KDM4E (0.44) HSD17B10COMTALDH1A1KDM4EGAA
SCHEMBL20176617 0.71 KMT2A (0.53) POLBHPGDNPSR1HSD17B10FAAH
SCHEMBL14827204 0.69 COMT (0.70) FAAHMGLLCOMTALDH1A1HSP90AA1
SCHEMBL21652820 0.69 NPSR1 (0.37) HPGDNPSR1HSD17B10COMTNPC1
SCHEMBL27858730 0.69 KMT2A (0.51) KMT2A
SCHEMBL2606749 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092047-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE JOINT STOCK COMPANY "BIOCAD" (RU) 2018-05-24 WO disclosed