SCHEMBL20176843

SCHEMBL20176843

CS(=O)(=O)NCCc1c(CCN)ccc2c1COC2=O

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 12/20 0.41
KCNH2 Q12809 7/20 0.41
NQO2 P16083 1/20 0.36
IMPDH2 P12268 1/20 0.35
IMPDH1 P20839 1/20 0.35
POLB P06746 1/20 0.34
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ALDH1A1 P00352 1/20 0.32
ALOX15 P16050 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
PRF1 P14222 1/20 0.32
ACHE P22303 1/20 0.32
SSTR1 P30872 1/20 0.32
SLC6A4 P31645 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20176799 0.74 KCNJ1 (0.68) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL20176945 0.71 KCNJ1 (0.46) KCNJ1KCNH2IMPDH2IMPDH1MAPT
SCHEMBL24135126 0.68 KCNJ1 (0.59) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL16836077 0.66 KCNJ1 (0.62) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL2729903 0.65 KCNJ1 (0.45) KCNJ1KCNH2MAPTKDM4EACHE
SCHEMBL2729380 0.64 KCNJ1 (0.44) KCNJ1KCNH2MAPTKDM4EACHE
SCHEMBL299969 0.62 KCNJ1 (0.44) KCNJ1KCNH2PRF1ACHESSTR1
SCHEMBL19433455 0.62 KCNJ1 (0.66) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL21243535 0.62 KCNJ1 (0.51) KCNJ1KCNH2ACHESSTR1SLC6A4
SCHEMBL21243537 0.62 KCNJ1 (0.51) KCNJ1KCNH2ACHESSTR1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018093569-A1 SUBSTITUTED BICYCLE HETEROCYCLIC DERIVATIVES USEFUL AS ROMK CHANNEL INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-24 WO disclosed