SCHEMBL20177498

SCHEMBL20177498

COc1cc(F)c([C@H]2Cc3nnc(C)n3C2)c(F)c1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
ADRA1A P35348 2/20 0.32
CPS1 P31327 1/20 0.31
LMNA P02545 1/20 0.31
BRD4 O60885 1/20 0.31
TAAR1 Q96RJ0 1/20 0.30
HCRTR1 O43613 1/20 0.30
HCRTR2 O43614 1/20 0.30
FPR2 P25090 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177493 0.76 ADRA1A (0.36) ADRA1ACPS1TAAR1HCRTR1HCRTR2
SCHEMBL20177558 0.74 GRM2 (0.45) LMNAFPR2
SCHEMBL20177825 0.73 ADRA1A (0.61) ADRA1A
SCHEMBL20177794 0.73 ADRA1A (0.61) ADRA1A
SCHEMBL18264318 0.72 FPR2 (0.34) TAAR1FPR2
SCHEMBL18264320 0.72 FPR2 (0.34) TAAR1FPR2
SCHEMBL19559537 0.70 HCRTR1 (0.38) CPS1HCRTR1HCRTR2FPR2
SCHEMBL19559422 0.70 HCRTR1 (0.38) CPS1HCRTR1HCRTR2FPR2
SCHEMBL18117769 0.69 PDE4A (0.50) CPS1BRD4HCRTR1HCRTR2
SCHEMBL19559459 0.69 PDE4A (0.50) CPS1BRD4HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed