SCHEMBL20177587

SCHEMBL20177587

COC1=NC[C@@H](c2c(F)cc(OC)cc2F)[C@@H]1NC(=O)OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
ACHE P22303 2/20 0.47
KCNQ2 O43526 1/20 0.46
FPR2 P25090 4/20 0.45
FPR1 P21462 2/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
CPB1 P15086 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
BRD4 O60885 2/20 0.39
BRD2 P25440 2/20 0.39
BRD3 Q15059 2/20 0.39
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16785452 0.89 FPR2 (0.49) CA1CA2ACHEKCNQ2FPR2
SCHEMBL16785365 0.87 FPR2 (0.50) CA1CA2ACHEKCNQ2FPR2
SCHEMBL20177608 0.84 FPR2 (0.46) CA1CA2ACHEKCNQ2FPR2
SCHEMBL20528327 0.82 FPR2 (0.44) CA1CA2ACHEKCNQ2FPR2
SCHEMBL18106440 0.80 FPR2 (0.68) FPR2FPR1
SCHEMBL29434207 0.80 FPR2 (0.68) FPR2FPR1
SCHEMBL18106745 0.80 CA1 (0.47) CA1CA2ACHEKCNQ2FPR2
SCHEMBL29434434 0.80 CA1 (0.47) CA1CA2ACHEKCNQ2FPR2
SCHEMBL16785438 0.80 FPR2 (0.68) FPR2FPR1
SCHEMBL18106743 0.80 CA1 (0.47) CA1CA2ACHEKCNQ2FPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed