SCHEMBL20177608

SCHEMBL20177608

COc1cc(F)c([C@@H]2CN=C(NCC(OC)OC)[C@H]2NC(=O)OCc2ccccc2)c(F)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 8/20 0.46
KCNQ2 O43526 1/20 0.45
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
ACHE P22303 1/20 0.42
FPR1 P21462 7/20 0.41
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
NAAA Q02083 2/20 0.36
BRD4 O60885 1/20 0.36
BRD2 P25440 1/20 0.36
BRD3 Q15059 1/20 0.36
CPB1 P15086 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177931 0.92 KCNQ2 (0.39) FPR2KCNQ2CA1CA2ACHE
SCHEMBL16785452 0.88 FPR2 (0.49) FPR2KCNQ2CA1CA2ACHE
SCHEMBL16785365 0.86 FPR2 (0.50) FPR2KCNQ2CA1CA2ACHE
SCHEMBL18264312 0.86 FPR2 (0.50) FPR2FPR1
SCHEMBL18264314 0.86 FPR2 (0.50) FPR2FPR1
SCHEMBL20177587 0.84 CA1 (0.47) FPR2KCNQ2CA1CA2ACHE
SCHEMBL20528327 0.81 FPR2 (0.44) FPR2KCNQ2CA1CA2ACHE
SCHEMBL16785438 0.77 FPR2 (0.68) FPR2FPR1
SCHEMBL29434207 0.77 FPR2 (0.68) FPR2FPR1
SCHEMBL18106440 0.77 FPR2 (0.68) FPR2FPR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed