SCHEMBL20177660

SCHEMBL20177660

CCOc1cc(F)c([C@@H]2CNC(=O)C2)c(F)c1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 12/20 0.49
FPR2 P25090 1/20 0.43
PDE4B Q07343 6/20 0.41
PDE4C Q08493 6/20 0.41
PDE4D Q08499 6/20 0.41
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
TSHR P16473 1/20 0.40
PIK3CD O00329 5/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19559432 1.00 PDE4A (0.49) PDE4AFPR2PDE4BPDE4CPDE4D
SCHEMBL16785337 0.84 PDE4A (0.49) PDE4AFPR2PDE4BPDE4CPDE4D
SCHEMBL19559455 0.84 PDE4A (0.49) PDE4AFPR2PDE4BPDE4CPDE4D
SCHEMBL20177904 0.83 FPR2 (0.39) PDE4AFPR2
SCHEMBL18117705 0.81 FPR1 (0.47) PDE4AFPR2PDE4BPDE4CPDE4D
SCHEMBL19559435 0.81 FPR1 (0.47) PDE4AFPR2PDE4BPDE4CPDE4D
SCHEMBL18590580 0.80 PDE4A (0.54) PDE4APDE4BPDE4CPDE4DMAOA
SCHEMBL19559407 0.80 PDE4A (0.54) PDE4APDE4BPDE4CPDE4DMAOA
SCHEMBL18590506 0.79 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL18590497 0.79 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed