SCHEMBL20179203

SCHEMBL20179203

CCOC(=O)c1ccc(CCCCC(=O)NOCc2ccc(OC(C)=O)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.47
CYP1A2 P05177 2/20 0.47
MEN1 O00255 1/20 0.47
SLC22A2 O15244 1/20 0.47
TMPRSS2 O15393 1/20 0.47
F2 P00734 1/20 0.47
F10 P00742 1/20 0.47
PLG P00747 1/20 0.47
F12 P00748 1/20 0.47
PLAU P00749 1/20 0.47
PLAT P00750 1/20 0.47
KLKB1 P03952 1/20 0.47
HPN P05981 1/20 0.47
CHRM2 P08172 1/20 0.47
CYP2D6 P10635 1/20 0.47
SLC6A2 P23975 1/20 0.47
SLC6A3 Q01959 1/20 0.47
KCNH2 Q12809 1/20 0.47
SLC47A2 Q86VL8 1/20 0.47
SLC47A1 Q96FL8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24023319 0.86 RXRA (0.41) KMT2AMEN1SMN1; SMN2NPC1CA1
SCHEMBL21578024 0.85 ELANE (0.42) KMT2ACYP1A2MEN1SLC22A2TMPRSS2
SCHEMBL21577995 0.82 HTT (0.39) KMT2ACYP1A2MEN1SLC22A2TMPRSS2
SCHEMBL20179151 0.82 FOLH1 (0.44) KMT2ACYP1A2MEN1SLC22A2TMPRSS2
SCHEMBL20179205 0.81 FOLH1 (0.52) KMT2ACYP1A2MEN1SLC22A2TMPRSS2
SCHEMBL20168306 0.79 FOLH1 (0.42) KMT2ACYP1A2MEN1SLC22A2TMPRSS2
SCHEMBL24023434 0.77 HDAC3 (0.44) LMNAMAPTSMN1; SMN2NPC1KDM4E
SCHEMBL24023430 0.76 ALDH1A1 (0.37) KMT2ASMN1; SMN2NPC1ALDH1A1RAB9A
SCHEMBL24023429 0.76 SLC7A5 (0.45) MAPTNPC1RAB9ACYP4F2CYP4A11
SCHEMBL1176935 0.76 CA12 (0.61) KMT2ACYP1A2MEN1SLC22A2TMPRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094334-A1 PRODRUGS OF HYDROXAMATE-BASED GCPII INHIBITORS THE JOHNS HOPKINS UNIVERSITY (US) 2018-05-24 WO disclosed