SCHEMBL2018052

SCHEMBL2018052

CS(=O)(=O)c1ccnc(Cl)n1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.38
GLP1R P43220 1/20 0.34
AURKA O14965 1/20 0.32
AURKB Q96GD4 1/20 0.32
CCR4 P51679 1/20 0.31
ABL1 P00519 1/20 0.31
BCR P11274 1/20 0.31
LMNA P02545 1/20 0.31
POLB P06746 1/20 0.31
LOX P28300 1/20 0.31
KDM4E B2RXH2 1/20 0.31
PKM P14618 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
RPS6KA5 O75582 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2047832 0.81 TDP1 (0.39) KDM4EPKMRPS6KA5
SCHEMBL30744221 0.80 TSHR (0.34) IDH1PTGS1PTGS2
SCHEMBL1750195 0.77 PARP1 (0.38) IDH1LMNAPOLBLOXKDM4E
SCHEMBL28686868 0.77 GRM4 (0.35) IDH1LMNAPOLBLOXKDM4E
SCHEMBL3599059 0.77 LOX (0.35) IDH1LMNAPOLBLOX
SCHEMBL3599060 0.75 ENPP2 (0.35) IDH1LMNAPOLBLOXKDM4E
SCHEMBL27841654 0.75 HDAC8 (0.33) IDH1LMNAPOLBLOX
SCHEMBL28938658 0.75 ROCK1 (0.45) AURKALMNAPOLB
SCHEMBL28022256 0.75 ALOX5AP (0.34) IDH1LMNAPOLBLOXPTGS1
SCHEMBL7068250 0.75 IDH1 (0.33) IDH1GLP1RLOX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5539088-A PROVIDE DYEINGS IN BRILLIANT SHADES WITH GOOD FASTNESS PROPERTIES AND HIGH DEGREE OF FIXATION HOECHST AKTIENGESELLSCHAFT (DE) 1996-07-23 US claimed
WO-2026041663-A1 P2X7 RECEPTOR ANTAGONISTS BREYE THERAPEUTICS APS (DK) 2026-02-26 WO disclosed
EP-4685141-A1 ISOINDOLINE DERIVATIVE, BENZOINDOLE DERIVATIVE AND USE THEREOF Shanghai Helioson Pharmaceutical Co., Ltd. (CN) 2026-01-28 EP disclosed
WO-2024193641-A1 ISOINDOLINE DERIVATIVE, BENZOINDOLE DERIVATIVE AND USE THEREOF 上海超阳药业有限公司 2024-09-26 WO disclosed
US-20240124406-A1 INHIBITORS OF TRANSCRIPTIONAL ENHANCED ASSOCIATE DOMAIN (TEAD) AND USES THEREOF DANA-FARBER CANCER INSTITUTE, INC. 2024-04-18 US disclosed
CN-117715906-A Glucagon-like peptide-1 receptor modulators and uses thereof 和博医药有限公司 2024-03-15 CN disclosed
CN-116761795-A Inhibitors of Transcription Enhancement Associated Domain (TEAD) and uses thereof 达纳-法伯癌症研究所股份有限公司 2023-09-15 CN disclosed
EP-4164752-A1 INHIBITORS OF TRANSCRIPTIONAL ENHANCED ASSOCIATE DOMAIN (TEAD) AND USES THEREOF Dana-Farber Cancer Institute, Inc. (US) 2023-04-19 EP disclosed
US-11512095-B2 BCL6 inhibitors THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL (GB) 2022-11-29 US disclosed
EP-2951169-B1 FLAP MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2019-08-28 EP disclosed
CN-1047778-C Pyrimido [5-4-d] pyrimidines, drugs containing these compounds, their use and process for preparing them THOMAE GMBH DR K (DE) 1999-12-29 CN disclosed
US-5770709-A BRILLIANT COLOR SHADES, GOOD FASTNESS DURING USE AT HIGH DEGREE OF FIXING DYSTAR TEXTILFARBEN GMBH & CO DEUTSCHLAND KG (DE) 1998-06-23 US disclosed
US-5539088-A PROVIDE DYEINGS IN BRILLIANT SHADES WITH GOOD FASTNESS PROPERTIES AND HIGH DEGREE OF FIXATION HOECHST AKTIENGESELLSCHAFT (DE) 1996-07-23 US disclosed
EP-0675172-A2 Water-solable azo compounds, process for their preparation and their use as dyestuffs HOECHST AKTIENGESELLSCHAFT (DE) 1995-10-04 EP disclosed
US-5197992-A Disazo dye, naphthol dye with triazole groups for wool, silk, polyamides and cellulose with triphenodioxazines IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-03-30 US disclosed
US-5196033-A BIS-azotriazinyl reactive dyes having an N-alkyl-phenylenediamine link for cellulose textiles IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-03-23 US disclosed
US-5059681-A BIS-AZOTRIAZINYL REACTIVE DYES HAVING AN N-ALKYL-PHENYLENEDIAMINE LINK IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-10-22 US disclosed
CN-1005738-B Printing method for cellulose fabric 西巴·盖尔基股份公司 1989-11-08 CN disclosed
EP-0256650-A2 Reactive dyes IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-02-24 EP disclosed
CN-85107872-A The printing method of cellulose fibre (fabric) 1986-07-09 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240124406-A1 INHIBITORS OF TRANSCRIPTIONAL ENHANCED ASSOCIATE DOMAIN (TEAD) AND USES THEREOF TEAD1, TEAD2, TEAD4 IDH1 876/4885GLP1R 4434/4885AURKA 3457/4885
US-11512095-B2 BCL6 inhibitors BCL6, BCL6B, BCL3 IDH1 602/4885GLP1R 1872/4885AURKA 2537/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.