SCHEMBL28022256

SCHEMBL28022256

CS(=O)(=O)c1ccnc(F)n1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
IDH1 O75874 1/20 0.33
LMNA P02545 1/20 0.31
POLB P06746 1/20 0.31
LOX P28300 1/20 0.31
MAPK1 P28482 1/20 0.31
GRM4 Q14833 1/20 0.31
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2044708 0.79 ALDH1A1 (0.38)
SCHEMBL3599059 0.77 LOX (0.35) ALOX5APFEN1IDH1LMNAPOLB
SCHEMBL28686868 0.77 GRM4 (0.35) ALOX5APFEN1IDH1LMNAPOLB
SCHEMBL1750195 0.77 PARP1 (0.38) ALOX5APFEN1IDH1LMNAPOLB
SCHEMBL3599060 0.75 ENPP2 (0.35) IDH1LMNAPOLBLOX
SCHEMBL28938658 0.75 ROCK1 (0.45) ALOX5APLMNAPOLB
SCHEMBL2018052 0.75 IDH1 (0.38) IDH1LMNAPOLBLOXPTGS1
SCHEMBL27841654 0.75 HDAC8 (0.33) IDH1LMNAPOLBLOX
SCHEMBL31475459 0.75 MALT1 (0.40) IDH1LMNAPOLBMAPK1PTGS2
SCHEMBL12417898 0.71 TGFBR1 (0.37) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104940202-B Inhibitors of influenza viruses replication 沃泰克斯药物股份有限公司 2018-10-16 CN disclosed
CN-104940202-A Inhibitors of influenza viruses replication VERTEX PHARMA 2015-09-30 CN disclosed
CN-104922128-A INHIBITORS OF INFLUENZA VIRUSES REPLICATION VERTEX PHARMA 2015-09-23 CN disclosed
CN-102458408-B Inhibitors of influenza virus replication VERTEX PHARMA 2015-06-03 CN disclosed