SCHEMBL20180754

SCHEMBL20180754

CCCc1cc(OC)c(N)c(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
CYP3A4 P08684 1/20 0.50
HTR2A P28223 2/20 0.48
HTR2C P28335 2/20 0.48
HTR2B P41595 2/20 0.48
CYP19A1 P11511 2/20 0.47
AOC3 Q16853 2/20 0.44
GABRA1 P14867 2/20 0.44
GABRB2 P47870 2/20 0.44
GABRA5 P31644 1/20 0.44
GABRA3 P34903 1/20 0.44
GABRA2 P47869 1/20 0.44
PTGS2 P35354 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ATM Q13315 1/20 0.42
HMGCR P04035 1/20 0.42
MAPT P10636 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27685436 0.82 PTGS2 (0.64) ALDH1A1HTR2AHTR2CHTR2BCYP19A1
SCHEMBL2500546 0.80 PTGS2 (0.68) ALDH1A1CYP3A4HTR2AHTR2CHTR2B
SCHEMBL5982004 0.79 ALDH1A1 (0.59) ALDH1A1CYP3A4HTR2AHTR2CHTR2B
SCHEMBL2442396 0.78 ALDH1A1 (0.50) ALDH1A1CYP3A4HTR2AHTR2CHTR2B
SCHEMBL223826 0.78 AKR1B1 (0.59) ALDH1A1CYP3A4GABRA1GABRB2GABRA5
SCHEMBL11060703 0.78 ALDH1A1 (0.50) ALDH1A1CYP3A4HTR2AHTR2CHTR2B
SCHEMBL13181141 0.78 ALDH1A1 (0.69) ALDH1A1CYP3A4CYP19A1AOC3GABRA1
SCHEMBL3362269 0.76 ALDH1A1 (0.45) ALDH1A1HTR2AHTR2CHTR2BCYP19A1
SCHEMBL3041350 0.75 AKR1B1 (0.61) ALDH1A1CYP3A4HMGCR
SCHEMBL31157855 0.75 PTGS2 (0.55) ALDH1A1CYP3A4HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018093579-A1 TRIAZOLE PHENYL COMPOUNDS AS AGONISTS OF THE APJ RECEPTOR AMGEN INC. (US) 2018-05-24 WO disclosed