SCHEMBL20181300

SCHEMBL20181300

C[C@@H](CC(=N)N)S(N)(=O)=O

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
BLM P54132 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TP53 P04637 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20181606 0.81 PMP22 (0.33) KDM4ECYP2D6CYP2C19BLMNPSR1
SCHEMBL28246970 0.78 ECE1 (0.32) BLMTP53CA1CA2CA9
SCHEMBL17337272 0.73 GABRP (0.41)
SCHEMBL10425679 0.71
SCHEMBL31511632 0.69
SCHEMBL18246035 0.69
SCHEMBL27159371 0.69
SCHEMBL28144836 0.68 TSHR (0.39) KDM4ECA1CA2CA9
SCHEMBL295045 0.68
SCHEMBL19641926 0.68 CA1 (0.38) TP53CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018093580-A1 TRIAZOLE PYRIDYL COMPOUNDS AS AGONISTS OF THE APJ RECEPTOR AMGEN INC. (US) 2018-05-24 WO disclosed