SCHEMBL2018150

SCHEMBL2018150

OCCc1ccnc(Cl)n1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.35
FFAR1 O14842 1/20 0.35
SORD Q00796 2/20 0.34
TRPV3 Q8NET8 1/20 0.31
RPS6KA5 O75582 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24258924 0.85 KCNH2 (0.35) RECQLFFAR1SORDKCNH2
SCHEMBL15577831 0.83
SCHEMBL2013407 0.79 FFAR1 (0.32) FFAR1RPS6KA5KCNH2
SCHEMBL27621059 0.79 FFAR1 (0.32) FFAR1RPS6KA5KCNH2
SCHEMBL4263566 0.79 HRH1 (0.45) FFAR1
SCHEMBL4273110 0.77 SORD (0.42) SORD
SCHEMBL16178953 0.76 KCNH2 (0.46) KCNH2
SCHEMBL6820237 0.76 CD274 (0.36) TRPV3
SCHEMBL27413913 0.76 KDM4E (0.35) FFAR1
SCHEMBL501903 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117659020-A Imidazo [1,2-b ] pyridazine derivative, and preparation method and application thereof 苏州朗睿生物医药有限公司 2024-03-08 CN disclosed
WO-2020081999-A1 ANDROGEN RECEPTOR MODULATORS AND METHODS FOR THEIR USE ESSA PHARMA, INC. (CA) 2020-04-23 WO disclosed
EP-2863914-A1 PYRAZOLYL DERIVATIVES AS SYK INHIBITORS Merck Sharp & Dohme Corp. (US) 2015-04-29 EP disclosed
WO-2013192125-A1 PYRAZOLYL DERIVATIVES AS SYK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-12-27 WO disclosed
EP-2513098-A1 AMINOPYRIMIDINES AS SYK INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-10-24 EP disclosed
WO-2011075515-A1 AMINOPYRIMIDINES AS SYK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-06-23 WO disclosed
WO-2011075517-A1 AMINOPYRIMIDINES AS SYK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-06-23 WO disclosed