SCHEMBL20181884

SCHEMBL20181884

C#CC(CC)n1cc(C)c2c(N)ncnc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.39
ADORA1 P30542 4/20 0.39
ADORA2B P29275 3/20 0.39
ADK P55263 1/20 0.38
SRC P12931 5/20 0.36
KDR P35968 5/20 0.36
LCK P06239 3/20 0.36
TEK Q02763 3/20 0.36
ABL1 P00519 3/20 0.36
EGFR P00533 3/20 0.36
PI4KB Q9UBF8 3/20 0.36
PIK3CD O00329 2/20 0.36
PIK3CA P42336 2/20 0.36
PIK3CB P42338 2/20 0.36
PIK3CG P48736 2/20 0.36
PRKDC P78527 2/20 0.36
HCK P08631 1/20 0.36
MTOR P42345 1/20 0.36
EPHB4 P54760 1/20 0.36
LRRK2 Q5S007 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20162958 0.85 MAP4K4 (0.44) ADORA2AADORA1ADORA2BADKSRC
SCHEMBL20182230 0.84 ADK (0.38) ADK
SCHEMBL20181879 0.82 RET (0.41) ADORA2AADORA1ADORA2BADKSRC
SCHEMBL19775103 0.80 ADORA2A (0.56) ADORA2AADORA1ADORA2BADKSRC
SCHEMBL20182185 0.76 RET (0.41) ADKSRCKDRLCKABL1
SCHEMBL2618932 0.76 PIK3CD (0.52) ADORA2AADORA1ADORA2BADKSRC
SCHEMBL30892143 0.75 ADORA2A (0.40) ADORA2AADORA1ADORA2BADKPI4KB
SCHEMBL24458478 0.73 RET (0.54) ADORA2AADORA1ADORA2BADKSRC
SCHEMBL20263231 0.72 RET (0.42) ADKSRCKDRLCKABL1
SCHEMBL20162872 0.72 ADK (0.39) ADK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed