SCHEMBL20182185

SCHEMBL20182185

C#CC(C1CC1)n1cc(C)c2c(N)ncnc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 14/20 0.41
LCK P06239 3/20 0.41
DAPK3 O43293 1/20 0.41
MAP4K4 O95819 1/20 0.41
PAK4 O96013 1/20 0.41
ABL1 P00519 1/20 0.41
FYN P06241 1/20 0.41
CSF1R P07333 1/20 0.41
IGF1R P08069 1/20 0.41
FGFR1 P11362 1/20 0.41
PRKACA P17612 1/20 0.41
FLT1 P17948 1/20 0.41
LTK P29376 1/20 0.41
KDR P35968 1/20 0.41
MAP2K2 P36507 1/20 0.41
FLT3 P36888 1/20 0.41
MAPK8 P45983 1/20 0.41
CSNK1A1 P48729 1/20 0.41
CDK8 P49336 1/20 0.41
CLK2 P49760 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20163009 0.85 MTOR (0.42) RETLCKDAPK3MAP4K4PAK4
SCHEMBL20181850 0.85 ADK (0.39) ADK
SCHEMBL20181879 0.80 RET (0.41) RETLCKDAPK3MAP4K4PAK4
SCHEMBL20181884 0.76 ADORA2A (0.39) RETLCKDAPK3MAP4K4PAK4
SCHEMBL30892155 0.75 DAPK3 (0.36) RETLCKDAPK3MAP4K4PAK4
SCHEMBL2618932 0.74 PIK3CD (0.52) RETLCKKDRADKSRC
SCHEMBL20162624 0.72 ADK (0.39) ADK
SCHEMBL24458478 0.71 RET (0.54) RETLCKABL1KDRDYRK1A
SCHEMBL19775103 0.70 ADORA2A (0.56) RETLCKABL1KDRADK
SCHEMBL24072104 0.69 RIPK2 (0.61) RETLCKDAPK3MAP4K4PAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed