SCHEMBL20181886

SCHEMBL20181886

CCC(c1ccccc1Cl)C(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.44
ADRB1 P08588 2/20 0.44
AOC3 Q16853 1/20 0.44
NISCH Q9Y2I1 1/20 0.43
TSHR P16473 3/20 0.41
HIF1A Q16665 3/20 0.40
CYP2D6 P10635 2/20 0.40
NFKB1 P19838 2/20 0.40
CYP3A4 P08684 2/20 0.39
CYP1A2 P05177 1/20 0.39
PNMT P11086 1/20 0.39
BLM P54132 2/20 0.39
LMNA P02545 2/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
CASP1 P29466 1/20 0.38
TAAR1 Q96RJ0 1/20 0.36
MC4R P32245 1/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20706300 0.84 ADRB2 (0.50) ADRB2ADRB1AOC3NISCHTSHR
SCHEMBL17755100 0.81 ADRB2 (0.40) ADRB2ADRB1AOC3NISCHHIF1A
SCHEMBL19518928 0.78 TSHR (0.59) ADRB2ADRB1AOC3NISCHTSHR
SCHEMBL17790152 0.78 TSHR (0.59) ADRB2ADRB1AOC3NISCHTSHR
SCHEMBL3789761 0.78 TSHR (0.59) ADRB2ADRB1AOC3NISCHTSHR
SCHEMBL17755097 0.77 ADRB2 (0.40) ADRB2ADRB1AOC3NISCHTSHR
SCHEMBL12120635 0.77 ADRB2 (0.40) ADRB2ADRB1AOC3NISCHTSHR
SCHEMBL2696923 0.77 TSHR (0.42) ADRB2ADRB1TSHRCYP2D6CYP3A4
SCHEMBL6643908 0.77 NISCH (0.44) ADRB2ADRB1AOC3NISCHTSHR
SCHEMBL18925051 0.76 TP53 (0.55) CYP3A4CYP1A2LMNAIDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11008339-B2 Substituted pyrazole compounds containing pyrimidine and preparation method and use thereof SHENYANG SINOCHEM AGROCHEMICALS R&D CO., LTD. (CN) 2021-05-18 US disclosed
US-20210015100-A1 SUBSTITUTED PYRIMIDINE COMPOUND AND PREPARATION METHOD AND USE THEREOF SHENYANG SINOCHEM AGROCHEMICALS R&D CO., LTD. (CN) 2021-01-21 US disclosed
US-20180141961-A1 Substituted Pyrazole Compounds Containing Pyrimidine and Preparation Method and Use Thereof SHENYANG SINOCHEM AGROCHEMICALS R&D CO., LTD. (CN) 2018-05-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210015100-A1 SUBSTITUTED PYRIMIDINE COMPOUND AND PREPARATION METHOD AND USE THEREOF GART, BROX, APRT ADRB2 2650/4885ADRB1 1626/4885AOC3 309/4885
US-20180141961-A1 Substituted Pyrazole Compounds Containing Pyrimidine and Preparation Method and Use Thereof APRT, GART, PNP ADRB2 1413/4885ADRB1 1100/4885AOC3 124/4885
US-11008339-B2 Substituted pyrazole compounds containing pyrimidine and preparation method and use thereof APRT, GART, PNP ADRB2 1413/4885ADRB1 1100/4885AOC3 124/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.