SCHEMBL20181956

SCHEMBL20181956

CCCCC(C)(CCCC)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC2 Q92769 1/20 0.48
EPHX2 P34913 2/20 0.40
NR1H4 Q96RI1 1/20 0.40
TRPV1 Q8NER1 2/20 0.40
TSHR P16473 1/20 0.40
LMNA P02545 1/20 0.39
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
CCR6 P51684 2/20 0.38
NOS3 P29474 2/20 0.38
NOS1 P29475 2/20 0.38
NOS2 P35228 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KIF11 P52732 1/20 0.38
PDE2A O00408 1/20 0.37
POLB P06746 1/20 0.37
KDM1A O60341 1/20 0.37
RCOR1 Q9UKL0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22024180 0.93 HDAC3 (0.46) HDAC3HDAC1HDAC2EPHX2NR1H4
SCHEMBL21549391 0.92 HDAC3 (0.45) HDAC3HDAC1HDAC2EPHX2NR1H4
SCHEMBL22024859 0.86 HDAC3 (0.48) HDAC3HDAC1HDAC2EPHX2NR1H4
SCHEMBL20866437 0.83 HDAC3 (0.41) HDAC3HDAC1HDAC2EPHX2NR1H4
SCHEMBL12700338 0.80 HDAC3 (0.46) HDAC3HDAC1HDAC2EPHX2NR1H4
SCHEMBL19965713 0.79 HDAC3 (0.43) HDAC3HDAC1HDAC2EPHX2NR1H4
SCHEMBL25622565 0.79 CNR2 (0.35) HDAC3HDAC1HDAC2ESR1ESR2
SCHEMBL2056145 0.76 LTA4H (0.52) HDAC3HDAC1HDAC2TSHRL3MBTL1
SCHEMBL17552746 0.74 NPC1 (0.55) HDAC3HDAC1HDAC2EPHX2NR1H4
SCHEMBL20313083 0.74 CNR2 (0.46) HDAC3HDAC1HDAC2TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11198693-B2 Functionalized heterocycles as antiviral agents ENANTA PHARMACEUTICALS, INC. (US) 2021-12-14 US disclosed
US-11008339-B2 Substituted pyrazole compounds containing pyrimidine and preparation method and use thereof SHENYANG SINOCHEM AGROCHEMICALS R&D CO., LTD. (CN) 2021-05-18 US disclosed
US-20200165249-A1 FUNCTIONALIZED HETEROCYCLES AS ANTIVIRAL AGENTS ENANTA PHARMACEUTICALS, INC. 2020-05-28 US disclosed
US-20180141961-A1 Substituted Pyrazole Compounds Containing Pyrimidine and Preparation Method and Use Thereof SHENYANG SINOCHEM AGROCHEMICALS R&D CO., LTD. (CN) 2018-05-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180141961-A1 Substituted Pyrazole Compounds Containing Pyrimidine and Preparation Method and Use Thereof APRT, GART, PNP HDAC3 2352/4885HDAC1 1322/4885HDAC2 595/4885
US-11008339-B2 Substituted pyrazole compounds containing pyrimidine and preparation method and use thereof APRT, GART, PNP HDAC3 2352/4885HDAC1 1322/4885HDAC2 595/4885
US-11198693-B2 Functionalized heterocycles as antiviral agents HCCS, HAVCR2, HDGF HDAC3 786/4885HDAC1 519/4885HDAC2 1540/4885
US-20200165249-A1 FUNCTIONALIZED HETEROCYCLES AS ANTIVIRAL AGENTS HCCS, HAVCR2, HDGF HDAC3 786/4885HDAC1 519/4885HDAC2 1540/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.