SCHEMBL20182227

SCHEMBL20182227

CCC(/C(=C/Nc1ccccc1F)N=N)n1cc(-c2nccnc2OC)c2c(N)ncnc21

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.36
SRC P12931 4/20 0.35
EIF2AK3 Q9NZJ5 1/20 0.34
KDR P35968 7/20 0.33
TEK Q02763 5/20 0.33
ABL1 P00519 4/20 0.33
ABL2 P42684 4/20 0.33
LCK P06239 2/20 0.33
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
PRKDC P78527 1/20 0.32
RET P07949 2/20 0.32
NEK7 Q8TDX7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20181916 0.87 CFTR (0.39) EGFRSRCEIF2AK3KDRTEK
SCHEMBL20182194 0.87 EIF2AK3 (0.36) EGFRSRCEIF2AK3KDRTEK
SCHEMBL20182248 0.83 LRRK2 (0.34) EGFRSRCEIF2AK3KDRTEK
SCHEMBL20181912 0.83 SRC (0.41) EGFRSRCEIF2AK3KDRTEK
SCHEMBL20182255 0.82 SRC (0.39) EGFRSRCEIF2AK3KDRTEK
SCHEMBL20182197 0.82 CFTR (0.43) EGFRSRCEIF2AK3KDRTEK
SCHEMBL20182198 0.81 SRC (0.34) EGFRSRCEIF2AK3KDRTEK
SCHEMBL20182274 0.81 EIF2AK3 (0.40) EGFRSRCEIF2AK3KDRTEK
SCHEMBL20182292 0.81 NEK7 (0.37) EGFRSRCEIF2AK3KDRTEK
SCHEMBL20182204 0.81 KDR (0.37) EGFRSRCEIF2AK3KDRTEK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed