SCHEMBL20181916

SCHEMBL20181916

CCC(/C(=C/Nc1ccccc1F)N=N)n1cc(-c2cncnc2OC)c2c(N)ncnc21

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.39
EGFR P00533 4/20 0.36
EIF2AK3 Q9NZJ5 4/20 0.35
SRC P12931 5/20 0.33
KDR P35968 4/20 0.33
ABL1 P00519 3/20 0.33
ABL2 P42684 3/20 0.33
TEK Q02763 3/20 0.33
LCK P06239 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20182265 0.92 NTRK1 (0.36) CFTREGFREIF2AK3KDRABL1
SCHEMBL20182194 0.91 EIF2AK3 (0.36) CFTREGFREIF2AK3SRCKDR
SCHEMBL20182224 0.90 EGFR (0.39) CFTREGFRSRCKDRABL1
SCHEMBL20182271 0.89 CFTR (0.35) CFTREGFREIF2AK3SRCKDR
SCHEMBL20182191 0.89 ALK (0.34) CFTREGFREIF2AK3SRCKDR
SCHEMBL20182227 0.87 EGFR (0.36) EGFREIF2AK3SRCKDRABL1
SCHEMBL20181906 0.87 EIF2AK3 (0.34) CFTREGFREIF2AK3SRCKDR
SCHEMBL20182289 0.84 NTRK1 (0.36) EGFREIF2AK3SRCKDRABL1
SCHEMBL20182235 0.84 EIF2AK3 (0.34) EGFREIF2AK3SRCKDRABL1
SCHEMBL20182198 0.84 SRC (0.34) CFTREGFREIF2AK3SRCKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed