SCHEMBL20182279

SCHEMBL20182279

CC(C)N/C=C(\C=N)Cn1c(Br)c(-c2ccc(Cl)cc2)c2c(N)ncnc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 5/20 0.39
RPS6KA3 P51812 5/20 0.36
KDR P35968 5/20 0.36
LCK P06239 4/20 0.36
TEK Q02763 4/20 0.36
CYP1A2 P05177 2/20 0.36
MEN1 O00255 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
SRC P12931 5/20 0.35
BTK Q06187 3/20 0.35
YES1 P07947 2/20 0.35
LYN P07948 2/20 0.35
BLK P51451 2/20 0.35
ABL1 P00519 2/20 0.35
DAPK3 O43293 1/20 0.35
RIPK2 O43353 1/20 0.35
EGFR P00533 1/20 0.35
HCK P08631 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20182223 0.87 RPS6KA3 (0.40) FYNRPS6KA3KDRLCKTEK
SCHEMBL20182205 0.80 SRC (0.47) FYNKDRLCKTEKSRC
SCHEMBL20182360 0.71 FYN (0.35) FYNRPS6KA3KDRLCKTEK
SCHEMBL20162990 0.71 FYN (0.41) FYNRPS6KA3KDRLCKTEK
SCHEMBL30355044 0.71 CYP1A2 (0.41) FYNRPS6KA3KDRLCKTEK
SCHEMBL20162800 0.71 CYP1A2 (0.41) FYNRPS6KA3KDRLCKTEK
SCHEMBL20162797 0.69 CYP1A2 (0.40) FYNRPS6KA3KDRLCKTEK
SCHEMBL13020205 0.66 CYP1A2 (0.47) FYNRPS6KA3KDRLCKTEK
SCHEMBL20182252 0.65 KDR (0.43) FYNKDRLCKTEKCYP1A2
SCHEMBL14682623 0.65 RPS6KA3 (0.54) FYNRPS6KA3KDRLCKTEK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed