SCHEMBL20182284

SCHEMBL20182284

Cc1cccc(N/C=C(\N=N)C(C)n2cc(-c3ccc(Cl)cc3)c3c(N)ncnc32)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.44
PIK3CA P42336 1/20 0.44
PIK3CB P42338 1/20 0.44
PIK3CG P48736 1/20 0.44
PRKDC P78527 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
KDR P35968 10/20 0.43
TEK Q02763 9/20 0.43
SRC P12931 7/20 0.43
LCK P06239 6/20 0.43
PDGFRB P09619 1/20 0.41
BTK Q06187 3/20 0.41
AURKA O14965 1/20 0.39
IKBKE Q14164 1/20 0.39
AURKB Q96GD4 1/20 0.39
FLT3 P36888 2/20 0.39
KIT P10721 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20182364 0.79 SRC (0.41) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL20181912 0.76 SRC (0.41) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL20182241 0.74 KDR (0.46) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL20182228 0.73 KDR (0.45) KDRTEKSRCLCKBTK
SCHEMBL13020100 0.72 KDR (0.68) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL20182362 0.72 CFTR (0.40) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL20181890 0.71 KDR (0.44) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL20181882 0.71 EGFR (0.42) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL20181883 0.71 NTRK1 (0.40) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL20162809 0.70 KDR (0.45) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed