SCHEMBL20184458

SCHEMBL20184458

O=C(O)c1c[nH]c2ncnc(-c3cccc(F)c3)c12

nearest known ligand 0.71

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 18/20 0.71
JAK2 O60674 11/20 0.71
ROCK2 O75116 1/20 0.52
LIMK1 P53667 1/20 0.52
KMO O15229 1/20 0.50
JAK1 P23458 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20184692 0.86 JAK3 (0.70) JAK3JAK2JAK1
SCHEMBL20184531 0.86 JAK3 (0.56) JAK3JAK2JAK1
SCHEMBL20184432 0.85 JAK3 (0.68) JAK3JAK2ROCK2LIMK1
SCHEMBL20184353 0.85 JAK3 (0.55) JAK3JAK2ROCK2LIMK1JAK1
SCHEMBL20184721 0.85 JAK3 (0.73) JAK3JAK2JAK1
SCHEMBL20184385 0.85 JAK3 (0.71) JAK3JAK2KMOJAK1
SCHEMBL20184686 0.84 JAK3 (0.55) JAK3JAK2ROCK2LIMK1
SCHEMBL15032692 0.83 JAK3 (1.00) JAK3JAK2JAK1
SCHEMBL20184454 0.83 JAK3 (0.70) JAK3JAK2ROCK2LIMK1
SCHEMBL20184488 0.82 JAK3 (0.50) JAK3JAK2ROCK2LIMK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2788000-B1 PYRROLOPYRIMIDINES AS JANUS KINASE INHIBITORS MERCK SHARP & DOHME (US) 2018-05-30 EP claimed