SCHEMBL20187568

SCHEMBL20187568

CC(=O)c1cc2c(o1)C(=O)c1c(O)cccc1C2=O

nearest known ligand 0.92

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 5/20 0.92
ALDH1A1 P00352 4/20 0.70
MAOA P21397 3/20 0.53
MAPT P10636 3/20 0.53
TSHR P16473 3/20 0.53
TDP1 Q9NUW8 3/20 0.53
MAPK1 P28482 2/20 0.53
LMNA P02545 2/20 0.53
HPGD P15428 2/20 0.53
ALOX15 P16050 2/20 0.53
MAOB P27338 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
HSD17B10 Q99714 2/20 0.53
HTT P42858 1/20 0.53
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
ELANE P08246 4/20 0.49
KDM4E B2RXH2 2/20 0.49
CYP3A4 P08684 2/20 0.49
RECQL P46063 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1450113 0.96 STAT3 (1.00) STAT3ALDH1A1MAOAMAPTTSHR
Napabucasin SCHEMBL29349770 0.83 STAT3 (1.00) STAT3ALDH1A1MAOAMAPTMAPK1
Napabucasin SCHEMBL1883845 0.83 STAT3 (1.00) STAT3ALDH1A1MAOAMAPTMAPK1
SCHEMBL10037450 0.83 STAT3 (0.77) STAT3ALDH1A1MAOAMAPTTSHR
SCHEMBL20187648 0.82 STAT3 (0.65) STAT3ALDH1A1MAPTTDP1LMNA
SCHEMBL7678888 0.81 STAT3 (0.61) STAT3ALDH1A1MAOAMAPTTSHR
SCHEMBL20190492 0.81 STAT3 (0.61) STAT3ALDH1A1MAOAMAPTTDP1
SCHEMBL20187596 0.80 STAT3 (0.60) STAT3ALDH1A1MAOAMAPTTSHR
SCHEMBL10037451 0.80 STAT3 (0.71) STAT3ALDH1A1MAOAMAPTTSHR
SCHEMBL20188858 0.78 STAT3 (0.65) STAT3ALDH1A1MAOAMAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018096401-A1 NEW NAPHTHO[2,3-B]FURAN DERIVATIVES BAN HITOSHI (JP) 2018-05-31 WO claimed
WO-2018096401-A1 NEW NAPHTHO[2,3-B]FURAN DERIVATIVES BAN HITOSHI (JP) 2018-05-31 WO disclosed