SCHEMBL20188248

SCHEMBL20188248

COc1cccc(NC(=O)c2ccc(Nc3ncc(SC)c(-c4cccnc4F)n3)cc2)c1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AURKA O14965 5/20 0.60
PTK2 Q05397 1/20 0.51
SMN1; SMN2 Q16637 2/20 0.50
TSHR P16473 1/20 0.50
NPC1 O15118 4/20 0.47
RAB9A P51151 4/20 0.47
ALDH1A1 P00352 2/20 0.47
KMT2A Q03164 2/20 0.47
TP53 P04637 1/20 0.47
PKM P14618 1/20 0.47
BTK Q06187 2/20 0.47
LCK P06239 1/20 0.47
CCNT1 O60563 1/20 0.46
CCNE1 P24864 1/20 0.46
CDK2 P24941 1/20 0.46
CDK9 P50750 1/20 0.46
KDR P35968 1/20 0.46
NLRP3 Q96P20 1/20 0.45
EGFR P00533 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20188707 0.88 AURKA (0.47) AURKAPTK2CCNT1CDK2CDK9
SCHEMBL20188200 0.88 AURKA (0.53) AURKAKMT2A
SCHEMBL30114845 0.88 AURKA (0.53) AURKAKMT2A
SCHEMBL20188249 0.85 AURKA (0.59) AURKAPTK2SMN1; SMN2TSHRKMT2A
SCHEMBL30114850 0.85 AURKA (0.45) AURKA
SCHEMBL20187976 0.85 AURKA (0.45) AURKA
SCHEMBL20188007 0.84 AURKA (0.45) AURKA
SCHEMBL20188270 0.83
SCHEMBL30114704 0.83
SCHEMBL21799092 0.82 TRPV1 (0.51) AURKANPC1RAB9AALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3544685-A1 HETROARYLAMINE COMPOUNDS FOR MODULATING THE HEDGEHOG PATHWAY AND PREPARING METHOD AND USES THEREOF Development Center for Biotechnology (TW) 2019-10-02 EP disclosed
WO-2018098250-A1 HETROARYLAMINE COMPOUNDS FOR MODULATING THE HEDGEHOG PATHWAY AND PREPARING METHOD AND USES THEREOF DEVELOPMENT CENTER FOR BIOTECHNOLOGY (TW) 2018-05-31 WO disclosed