SCHEMBL20188249

SCHEMBL20188249

COc1ccccc1NC(=O)c1ccc(Nc2ncc(SC)c(-c3cccnc3F)n2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 7/20 0.59
PTK2 Q05397 3/20 0.51
JAK2 O60674 1/20 0.51
NTRK1 P04629 1/20 0.51
TYK2 P29597 1/20 0.51
KDR P35968 1/20 0.51
JAK3 P52333 1/20 0.51
PTK2B Q14289 1/20 0.51
NTRK3 Q16288 1/20 0.51
NTRK2 Q16620 1/20 0.51
MAPT P10636 2/20 0.49
MEN1 O00255 1/20 0.45
AHR P35869 1/20 0.45
KMT2A Q03164 1/20 0.45
MLYCD O95822 1/20 0.45
TSHR P16473 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PRKCA P17252 1/20 0.44
P4HTM Q9NXG6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20188707 0.90 AURKA (0.47) AURKAPTK2JAK2NTRK1TYK2
SCHEMBL30114784 0.89 AURKA (0.58) AURKAMAPTCDK2AURKB
SCHEMBL20188503 0.89 AURKA (0.58) AURKAMAPTCDK2AURKB
SCHEMBL20187976 0.87 AURKA (0.45) AURKA
SCHEMBL30114850 0.87 AURKA (0.45) AURKA
SCHEMBL30114845 0.86 AURKA (0.53) AURKAMEN1KMT2ANAMPT
SCHEMBL20188200 0.86 AURKA (0.53) AURKAMEN1KMT2ANAMPT
SCHEMBL20188248 0.85 AURKA (0.60) AURKAPTK2KDRKMT2ATSHR
SCHEMBL20188007 0.83 AURKA (0.45) AURKA
SCHEMBL20188270 0.82

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3544685-A1 HETROARYLAMINE COMPOUNDS FOR MODULATING THE HEDGEHOG PATHWAY AND PREPARING METHOD AND USES THEREOF Development Center for Biotechnology (TW) 2019-10-02 EP disclosed
WO-2018098250-A1 HETROARYLAMINE COMPOUNDS FOR MODULATING THE HEDGEHOG PATHWAY AND PREPARING METHOD AND USES THEREOF DEVELOPMENT CENTER FOR BIOTECHNOLOGY (TW) 2018-05-31 WO disclosed