SCHEMBL30114845

SCHEMBL30114845

CSc1cnc(Nc2ccc(C(=O)Nc3ccccc3)cc2)nc1-c1cccnc1F

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AURKA O14965 10/20 0.53
BRD4 O60885 1/20 0.48
NAMPT P43490 1/20 0.46
MEN1 O00255 1/20 0.46
POLB P06746 1/20 0.46
KMT2A Q03164 1/20 0.46
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
TRPV1 Q8NER1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20188200 1.00 AURKA (0.53) AURKABRD4NAMPTMEN1POLB
SCHEMBL21799092 0.90 TRPV1 (0.51) AURKAMEN1POLBKMT2AGSK3A
SCHEMBL30114784 0.89 AURKA (0.58) AURKA
SCHEMBL20188503 0.89 AURKA (0.58) AURKA
SCHEMBL20188007 0.89 AURKA (0.45) AURKA
SCHEMBL20188270 0.88
SCHEMBL30114704 0.88
SCHEMBL20188248 0.88 AURKA (0.60) AURKAKMT2A
SCHEMBL20188249 0.86 AURKA (0.59) AURKANAMPTMEN1KMT2A
SCHEMBL30114720 0.86 CDK2 (0.52) AURKAGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110139692-B Heteroaryl amine compounds for modulating hedgehog pathway and methods of making and using the same 财团法人生物技术开发中心 2023-08-25 CN claimed
CN-110139692-B Heteroaryl amine compounds for modulating hedgehog pathway and methods of making and using the same 财团法人生物技术开发中心 2023-08-25 CN disclosed