SCHEMBL20190260

SCHEMBL20190260

CSc1cnc(Nc2ccc(C(=O)Nc3cc(C)ccc3C)cc2)nc1-c1ccc(F)cc1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AURKA O14965 3/20 0.48
ABL1 P00519 1/20 0.46
PDGFRB P09619 1/20 0.46
BCR P11274 1/20 0.46
PDGFRA P16234 1/20 0.46
TP53 P04637 1/20 0.45
MAPT P10636 1/20 0.45
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
KMT2A Q03164 1/20 0.44
KCNMA1 Q12791 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20188166 0.88 AURKA (0.44) AURKAABL1PDGFRBPDGFRA
SCHEMBL30530307 0.88 AURKA (0.44) AURKAABL1PDGFRBPDGFRA
SCHEMBL30114879 0.86 BCHE (0.46) AURKAABL1BCR
SCHEMBL20187744 0.86 BCHE (0.46) AURKAABL1BCR
SCHEMBL21799119 0.85
SCHEMBL20188725 0.84 MCHR1 (0.54) ABL1BCR
SCHEMBL30114741 0.84 MCHR1 (0.54) ABL1BCR
SCHEMBL30530294 0.84 ABL1 (0.54) ABL1PDGFRBBCRPDGFRA
SCHEMBL21799066 0.84 ABL1 (0.54) ABL1PDGFRBBCRPDGFRA
SCHEMBL21799072 0.83 RAB9A (0.51) AURKAABL1PDGFRBBCRPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3544685-A1 HETROARYLAMINE COMPOUNDS FOR MODULATING THE HEDGEHOG PATHWAY AND PREPARING METHOD AND USES THEREOF Development Center for Biotechnology (TW) 2019-10-02 EP disclosed
WO-2018098250-A1 HETROARYLAMINE COMPOUNDS FOR MODULATING THE HEDGEHOG PATHWAY AND PREPARING METHOD AND USES THEREOF DEVELOPMENT CENTER FOR BIOTECHNOLOGY (TW) 2018-05-31 WO disclosed