SCHEMBL20190908

SCHEMBL20190908

CCOc1ccc(-c2cc(Nc3ccc(C(=O)Nc4cc(CN5CCN(C)CC5)ccc4C)cc3)ncc2SC)c(OCC)c1OCC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 11/20 0.46
ABL1 P00519 9/20 0.44
BRAF P15056 6/20 0.44
KIT P10721 5/20 0.44
BCR P11274 4/20 0.44
PDGFRA P16234 3/20 0.44
ABL2 P42684 3/20 0.44
ERBB2 P04626 2/20 0.44
LCK P06239 2/20 0.44
FYN P06241 2/20 0.44
CSF1R P07333 2/20 0.44
LYN P07948 2/20 0.44
PDGFRB P09619 2/20 0.44
FGR P09769 2/20 0.44
SRC P12931 2/20 0.44
NQO2 P16083 2/20 0.44
EPHA8 P29322 2/20 0.44
FRK P42685 2/20 0.44
BLK P51451 2/20 0.44
DDR1 Q08345 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20188084 0.84 ABL1 (0.49) EGFRABL1BRAFKITBCR
SCHEMBL20188677 0.83 BRAF (0.49) EGFRABL1BRAFKITBCR
SCHEMBL30114739 0.82 ABL1 (0.47) EGFRABL1BRAFKITBCR
SCHEMBL21799087 0.82 ABL1 (0.47) EGFRABL1BRAFKITBCR
SCHEMBL30530293 0.77 RAB9A (0.53) ABL1BCRLMNAMAPK14F10
SCHEMBL21799076 0.77 RAB9A (0.53) ABL1BCRLMNAMAPK14F10
SCHEMBL20188790 0.75 ABL1 (0.51) ABL1BCRLMNAMAPK14
SCHEMBL21799066 0.74 ABL1 (0.54) EGFRABL1BRAFKITBCR
SCHEMBL30530294 0.74 ABL1 (0.54) EGFRABL1BRAFKITBCR
SCHEMBL20191064 0.73 ABL1 (0.52) EGFRABL1BRAFKITBCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3544685-A1 HETROARYLAMINE COMPOUNDS FOR MODULATING THE HEDGEHOG PATHWAY AND PREPARING METHOD AND USES THEREOF Development Center for Biotechnology (TW) 2019-10-02 EP disclosed
WO-2018098250-A1 HETROARYLAMINE COMPOUNDS FOR MODULATING THE HEDGEHOG PATHWAY AND PREPARING METHOD AND USES THEREOF DEVELOPMENT CENTER FOR BIOTECHNOLOGY (TW) 2018-05-31 WO disclosed