SCHEMBL20193704

SCHEMBL20193704

Cc1ccc([C@H](O)[C@@H](NC(=O)[C@@H]2CCCN2)c2ccccc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.52
CYP2D6 P10635 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2C19 P33261 1/20 0.52
CYP2C9 P11712 1/20 0.48
TSHR P16473 1/20 0.48
CTSC P53634 3/20 0.47
KEAP1 Q14145 2/20 0.42
NFE2L2 Q16236 2/20 0.42
GPR88 Q9GZN0 1/20 0.41
LMNA P02545 3/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TP53 P04637 1/20 0.39
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16139975 0.93 CYP3A4 (0.55) CYP3A4CYP2D6CYP1A2CYP2C19CYP2C9
SCHEMBL16376134 0.93 CYP3A4 (0.55) CYP3A4CYP2D6CYP1A2CYP2C19CYP2C9
SCHEMBL16015165 0.93 CYP3A4 (0.55) CYP3A4CYP2D6CYP1A2CYP2C19CYP2C9
SCHEMBL16015166 0.93 CYP3A4 (0.55) CYP3A4CYP2D6CYP1A2CYP2C19CYP2C9
SCHEMBL12333752 0.93 CYP3A4 (0.55) CYP3A4CYP2D6CYP1A2CYP2C19CYP2C9
SCHEMBL13974186 0.82 CYP3A4 (0.57) CYP3A4CYP2D6CYP1A2CYP2C19CYP2C9
SCHEMBL976838 0.77 RECQL (0.62) CYP3A4CYP2D6CYP1A2CYP2C19CYP2C9
SCHEMBL7313737 0.77 RECQL (0.62) CYP3A4CYP2D6CYP1A2CYP2C19CYP2C9
SCHEMBL7313727 0.77 RECQL (0.62) CYP3A4CYP2D6CYP1A2CYP2C19CYP2C9
SCHEMBL24056571 0.77 LMNA (0.60) CYP3A4CYP2D6CYP1A2CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9981935-B2 Formation of chiral 4-chromanones using chiral pyrrolidines in the presence of acids DSM IP ASSETS B.V. (NL) 2018-05-29 US disclosed