SCHEMBL20195261

SCHEMBL20195261

BC(O)(O)COc1ccc(Br)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
GABRA5 P31644 1/20 0.37
ALDH1A1 P00352 2/20 0.36
ADRA2A P08913 2/20 0.34
ADRA2B P18089 2/20 0.34
ADRA2C P18825 2/20 0.34
PLAU P00749 1/20 0.34
GBA1 P04062 1/20 0.34
DGAT1 O75907 1/20 0.34
THRB P10828 1/20 0.32
TSHR P16473 1/20 0.32
MAPT P10636 2/20 0.32
POLB P06746 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 3/20 0.31
NPC1 O15118 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
PKM P14618 1/20 0.31
FDPS P14324 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18402510 0.87 KDM4E (0.38) KDM4EL3MBTL1GABRA5ALDH1A1ADRA2A
SCHEMBL1403884 0.84 KDM4E (0.43) KDM4EL3MBTL1GABRA5ALDH1A1ADRA2A
SCHEMBL2461154 0.79 L3MBTL1 (0.56) KDM4EL3MBTL1GABRA5ALDH1A1THRB
SCHEMBL1821132 0.75 GBA1 (0.40) KDM4EL3MBTL1GABRA5ALDH1A1GBA1
SCHEMBL16787910 0.75 KDM4E (0.45) KDM4EL3MBTL1ALDH1A1DGAT1MAPT
SCHEMBL22031991 0.74 KDM4E (0.41) KDM4EGABRA5ALDH1A1GBA1DGAT1
SCHEMBL1284075 0.73 KDM4E (0.42) KDM4EGABRA5ALDH1A1ADRA2AADRA2B
SCHEMBL374769 0.73 DGAT1 (0.58) KDM4EL3MBTL1ALDH1A1DGAT1RAB9A
SCHEMBL30815211 0.72 KDM4E (0.41) KDM4EL3MBTL1GABRA5ALDH1A1ADRA2A
SCHEMBL156935 0.72 MAPT (0.52) KDM4EGABRA5ALDH1A1GBA1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2729447-B1 POSITIVE ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTOR H LUNDBECK AS (DK) 2018-05-30 EP disclosed