SCHEMBL20197186

SCHEMBL20197186

O=C(NC1CC1)c1cc(I)ccc1F

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.54
KDM1A O60341 4/20 0.53
MAOA P21397 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
TAS1R3 Q7RTX0 3/20 0.44
TAS1R1 Q7RTX1 3/20 0.44
TAS1R2 Q8TE23 3/20 0.44
CNR1 P21554 1/20 0.44
ALDH1A1 P00352 3/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
P2RX7 Q99572 1/20 0.43
GRM5 P41594 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
MAPK14 Q16539 1/20 0.42
TSHR P16473 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20197291 0.92 KDM1A (0.60) HPGDKDM1AMAOASMN1; SMN2NPC1
SCHEMBL3225623 0.87 HPGD (0.55) HPGDKDM1AMAOASMN1; SMN2NPC1
SCHEMBL7118324 0.82 NPC1 (0.51) HPGDNPC1RAB9ATAS1R3TAS1R1
SCHEMBL21516993 0.81 NPC1 (0.51) HPGDKDM1AMAOASMN1; SMN2NPC1
SCHEMBL20460485 0.81 NPC1 (0.55) HPGDKDM1AMAOASMN1; SMN2NPC1
SCHEMBL17373238 0.81 HPGD (0.58) HPGDSMN1; SMN2NPC1RAB9ATAS1R3
SCHEMBL16236985 0.81 HPGD (0.54) HPGDKDM1AMAOASMN1; SMN2NPC1
SCHEMBL16548437 0.81 TAS1R3 (0.58) HPGDKDM1AMAOASMN1; SMN2NPC1
SCHEMBL21090793 0.77 HPGD (0.48) HPGDNPC1RAB9ATAS1R3TAS1R1
SCHEMBL3233932 0.77 NPC1 (0.53) HPGDSMN1; SMN2NPC1RAB9ATAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3038622-B1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECH LLC (US) 2018-05-30 EP disclosed