SCHEMBL20197291

SCHEMBL20197291

O=C(NC1CCCCC1)c1cc(I)ccc1F

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.60
MAOA P21397 1/20 0.60
NPC1 O15118 9/20 0.57
RAB9A P51151 8/20 0.57
SMN1; SMN2 Q16637 5/20 0.57
ALDH1A1 P00352 5/20 0.50
HPGD P15428 2/20 0.50
LMNA P02545 2/20 0.50
KDM4E B2RXH2 1/20 0.50
HTT P42858 1/20 0.50
TSHR P16473 1/20 0.49
MAPT P10636 1/20 0.49
EPHX1 P07099 1/20 0.49
EPHX2 P34913 1/20 0.49
CNR1 P21554 2/20 0.47
CNR2 P34972 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20197186 0.92 HPGD (0.54) KDM1AMAOANPC1RAB9ASMN1; SMN2
SCHEMBL20460485 0.87 NPC1 (0.55) KDM1AMAOANPC1RAB9ASMN1; SMN2
SCHEMBL21516993 0.84 NPC1 (0.51) KDM1AMAOANPC1RAB9ASMN1; SMN2
SCHEMBL16548438 0.82 NPC1 (0.66) KDM1AMAOANPC1RAB9ASMN1; SMN2
SCHEMBL4574293 0.81 HPGD (0.64) NPC1RAB9ASMN1; SMN2HPGDLMNA
SCHEMBL6228759 0.81 NPC1 (0.63) NPC1RAB9ASMN1; SMN2ALDH1A1HPGD
SCHEMBL3225623 0.80 HPGD (0.55) KDM1AMAOANPC1RAB9ASMN1; SMN2
SCHEMBL13493618 0.80 KDM1A (0.57) KDM1AMAOANPC1RAB9ASMN1; SMN2
SCHEMBL29951948 0.80 KDM1A (0.57) KDM1AMAOANPC1RAB9ASMN1; SMN2
SCHEMBL16544524 0.79 KDM1A (0.56) KDM1AMAOANPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3038622-B1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECH LLC (US) 2018-05-30 EP disclosed