SCHEMBL20197278

SCHEMBL20197278

CCCc1nc(-c2nc(-c3ccc(NSC(F)(F)F)cc3Cl)cs2)no1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 16/20 0.39
CNR1 P21554 12/20 0.36
PGK1 P00558 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
HTT P42858 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
KDM4E B2RXH2 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16535265 0.85 CNR2 (0.39) CNR2CNR1PGK1NPC1RAB9A
SCHEMBL20197218 0.84 MAPT (0.36) NPC1RAB9ASMN1; SMN2LMNAMAPT
SCHEMBL20197297 0.83 CYP19A1 (0.35) NPC1RAB9ASMN1; SMN2LMNAMAPT
SCHEMBL20197472 0.83 CYP1B1 (0.36) NPC1RAB9ASMN1; SMN2HTTLMNA
SCHEMBL20197267 0.80 C1S (0.34) NPC1RAB9ASMN1; SMN2HTTLMNA
SCHEMBL20197221 0.80 SREBF2 (0.55) LMNAMAPTKDM4E
SCHEMBL20197220 0.79 SREBF2 (0.35) LMNAMAPTRXFP1KDM4E
SCHEMBL20197342 0.78 LMNA (0.37) NPC1RAB9ASMN1; SMN2HTTLMNA
SCHEMBL20197302 0.76 SMN1; SMN2 (0.46) NPC1RAB9ASMN1; SMN2HTTLMNA
SCHEMBL16548477 0.76 CNR2 (0.39) CNR2CNR1NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3038622-B1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECH LLC (US) 2018-05-30 EP disclosed