SCHEMBL20197302

SCHEMBL20197302

FC(F)(F)SNc1ccc(-c2csc(-c3ccccc3)n2)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.46
RAB9A P51151 5/20 0.46
KDM4E B2RXH2 5/20 0.46
NPC1 O15118 4/20 0.46
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
KMT2A Q03164 5/20 0.43
MEN1 O00255 4/20 0.43
CYP1A2 P05177 3/20 0.43
SMO Q99835 2/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 2/20 0.43
CYP2C19 P33261 1/20 0.43
MAPT P10636 4/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20197228 0.88 CYP1A1 (0.42) SMN1; SMN2RAB9AKDM4ENPC1CRHBP
SCHEMBL20197320 0.87 SREBF2 (0.44) SMN1; SMN2RAB9AKDM4ENPC1CRHBP
SCHEMBL20197309 0.83 CYP1B1 (0.41) SMN1; SMN2RAB9AKDM4ENPC1CRHBP
SCHEMBL20197240 0.82 ALDH1A1 (0.53) SMN1; SMN2RAB9AKDM4ENPC1KMT2A
SCHEMBL20197440 0.82 KDM4E (0.36) SMN1; SMN2RAB9AKDM4ENPC1CRHBP
SCHEMBL20197355 0.82 MEN1 (0.53) SMN1; SMN2RAB9AKDM4ENPC1KMT2A
SCHEMBL20197336 0.82 CYP19A1 (0.46) SMN1; SMN2RAB9AKDM4ENPC1CRHBP
SCHEMBL20197318 0.81 EIF4E (0.46) SMN1; SMN2RAB9AKDM4ENPC1CRHBP
SCHEMBL20197271 0.80 MEN1 (0.39) SMN1; SMN2RAB9AKDM4ENPC1KMT2A
SCHEMBL20197249 0.80 SREBF2 (0.43) KDM4EALDH1A1MAPTATMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3038622-B1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECH LLC (US) 2018-05-30 EP disclosed