SCHEMBL20197368

SCHEMBL20197368

[O-][S+](Nc1ccc(-c2csc(-c3ccnc(N4CCCCC4)c3)n2)c(Cl)c1)C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.35
SMG1 Q96Q15 3/20 0.34
ITGB2 P05107 2/20 0.34
ICAM1 P05362 2/20 0.34
ITGAL P20701 2/20 0.34
PIK3C3 Q8NEB9 1/20 0.34
MTOR P42345 2/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
CRHBP P24387 1/20 0.33
RAB9A P51151 1/20 0.33
CRHR2 Q13324 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CDK1 P06493 1/20 0.33
CDK2 P24941 1/20 0.33
EIF4E P06730 2/20 0.33
SREBF2 Q12772 1/20 0.33
CYP1B1 Q16678 2/20 0.33
CYP1A2 P05177 1/20 0.33
PIM1 P11309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20197238 0.85 CYP19A1 (0.44) KDM4ENPC1CRHBPRAB9ACRHR2
SCHEMBL16535259 0.82 SMG1 (0.39) MAPK14SMG1MTORKDM4ENPC1
SCHEMBL20197301 0.81 KDM4E (0.34) KDM4ENPC1CRHBPRAB9ACRHR2
SCHEMBL20197235 0.80 SREBF2 (0.42) KDM4ESREBF2
SCHEMBL20197223 0.79 SREBF2 (0.42) KDM4ESREBF2
SCHEMBL20197350 0.78 PIM1 (0.41) SMG1PIK3C3MTORKDM4ECDK2
SCHEMBL20197304 0.78 CDK2 (0.39) KDM4ENPC1CRHBPRAB9ACRHR2
SCHEMBL20197481 0.78 EIF4E (0.37) KDM4ENPC1CRHBPRAB9ACRHR2
SCHEMBL16536446 0.77 NMT1 (0.42) SMG1PIK3C3MTORKDM4ECDK2
SCHEMBL20197337 0.77 CYP1A2 (0.40) KDM4ENPC1CRHBPRAB9ACRHR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3038622-B1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECH LLC (US) 2018-05-30 EP disclosed