SCHEMBL20197304

SCHEMBL20197304

Nc1nccc(-c2nc(-c3ccc(N[S+]([O-])C(F)(F)F)cc3Cl)cs2)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 6/20 0.39
CDC7 O00311 5/20 0.39
CCNE1 P24864 5/20 0.39
DBF4 Q9UBU7 5/20 0.39
CCNT1 O60563 3/20 0.39
CDK9 P50750 3/20 0.39
KDM4E B2RXH2 3/20 0.39
CSNK2A2 P19784 2/20 0.39
CSNK1A1 P48729 2/20 0.39
CSNK1D P48730 2/20 0.39
CSNK2B P67870 2/20 0.39
CSNK2A1 P68400 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HSP90AA1 P07900 1/20 0.38
AMY1A P0DUB6 1/20 0.37
MALT1 Q9UDY8 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20197238 0.84 CYP19A1 (0.44) KDM4ENPC1RAB9AAMY1ACYP19A1
SCHEMBL16535320 0.80 CDC7 (0.39) CDK2CDC7CCNE1DBF4CCNT1
SCHEMBL20197159 0.80 CYP19A1 (0.33) KDM4ENPC1RAB9AAMY1ACYP19A1
SCHEMBL20197204 0.80 ATP4A (0.33) MAPT
SCHEMBL20197337 0.79 CYP1A2 (0.40) KDM4ENPC1RAB9AMAPTCYP19A1
SCHEMBL20197301 0.79 KDM4E (0.34) KDM4ENPC1RAB9AMAPTCYP19A1
SCHEMBL20197235 0.79 SREBF2 (0.42) KDM4EMAPTL3MBTL1ALDH1A1
SCHEMBL20197443 0.78 C1S (0.39) KDM4ENPC1RAB9AMAPTAMY1A
SCHEMBL20197223 0.78 SREBF2 (0.42) KDM4EMAPTL3MBTL1ALDH1A1
SCHEMBL20197368 0.78 MAPK14 (0.35) CDK2KDM4ENPC1RAB9ACYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3038622-B1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECH LLC (US) 2018-05-30 EP disclosed