SCHEMBL20200044

SCHEMBL20200044

O=C(O)CN1CCN(CC(=O)O)CCN(CC(=O)N(CC(=O)NCC(CNC(=O)CN(Cc2ccccc2)C(=O)CN2CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC2)(CNC(=O)CN(Cc2ccccc2)C(=O)CN2CCN(CC(=O)O)CCN(CC(O)O)CCN(CC(=O)O)CC2)NC(=O)CN(Cc2ccccc2)C(=O)CN2CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC2)Cc2ccccc2)CCN(CC(=O)O)CC1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.38
HDAC6 Q9UBN7 2/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 2/20 0.37
POLB P06746 1/20 0.37
FOLH1 Q04609 4/20 0.36
CTSS P25774 2/20 0.35
CTSK P43235 1/20 0.35
CTSL P07711 1/20 0.35
NPSR1 Q6W5P4 1/20 0.34
LMNA P02545 1/20 0.34
MCHR1 Q99705 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22112574 0.91 HDAC1 (0.39) HDAC1HDAC6MEN1KMT2AALDH1A1
SCHEMBL20200110 0.85 CACNA2D1 (0.36) HDAC1HDAC6MEN1KMT2AALDH1A1
SCHEMBL22069305 0.84 HDAC1 (0.42) HDAC1HDAC6MEN1KMT2AALDH1A1
SCHEMBL20199792 0.82
SCHEMBL20199838 0.80 HSD17B10 (0.33) ALDH1A1
SCHEMBL20200026 0.79
SCHEMBL22069430 0.79 MEN1 (0.40) HDAC1HDAC6MEN1KMT2AALDH1A1
SCHEMBL20199802 0.78 ALDH1A1 (0.34) ALDH1A1
SCHEMBL23656474 0.78 MEN1 (0.39) HDAC1HDAC6MEN1KMT2AALDH1A1
SCHEMBL20187486 0.75 ALDH1A1 (0.49) MEN1KMT2AALDH1A1POLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018096082-A1 HIGH RELAXIVITY GADOLINIUM CHELATE COMPOUNDS FOR USE IN MAGNETIC RESONANCE IMAGING BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-31 WO disclosed