SCHEMBL20199802

SCHEMBL20199802

O=C(O)CN1CCN(CC(=O)O)CCN(CC(=O)N(CC(=O)NCC(CNC(=O)CN(C(=O)CN2CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC2)C2CCCC2)(CNC(=O)CN(C(=O)CN2CCN(CC(=O)O)CCN(CC(O)O)CCN(CC(=O)O)CC2)C2CCCC2)NC(=O)CN(C(=O)CN2CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC2)C2CCCC2)C2CCCC2)CCN(CC(=O)O)CC1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
MAPK1 P28482 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HTT P42858 1/20 0.30
HSD11B1 P28845 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22112106 0.91 ALDH1A1 (0.35) ALDH1A1MAPK1HSD17B10HSD11B1
SCHEMBL22069326 0.83 ALDH1A1 (0.37) ALDH1A1MAPK1HSD17B10HSD11B1
SCHEMBL20199792 0.81
SCHEMBL20199838 0.78 HSD17B10 (0.33) ALDH1A1HSD17B10
SCHEMBL22069436 0.78 ALDH1A1 (0.32) ALDH1A1MAPK1HSD17B10HTT
SCHEMBL22403182 0.78
SCHEMBL20200044 0.78 HDAC1 (0.38) ALDH1A1
SCHEMBL20200026 0.78
SCHEMBL20200110 0.77 CACNA2D1 (0.36) ALDH1A1MAPK1HTT
SCHEMBL20200043 0.74 HSD11B1 (0.41) HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018096082-A1 HIGH RELAXIVITY GADOLINIUM CHELATE COMPOUNDS FOR USE IN MAGNETIC RESONANCE IMAGING BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-31 WO disclosed