SCHEMBL20200052

SCHEMBL20200052

COC(=O)CN1CCN(CC(=O)OC)CCN(CC(=O)N(C)CC(=O)O)CCN(CC(=O)OC)CC1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
POLB P06746 1/20 0.37
MVD P53602 1/20 0.36
SIGMAR1 Q99720 1/20 0.34
KDM4E B2RXH2 2/20 0.33
HTT P42858 1/20 0.33
DRD4 P21917 1/20 0.33
OPRM1 P35372 1/20 0.32
OPRL1 P41146 1/20 0.32
TACR1 P25103 1/20 0.32
TSHR P16473 1/20 0.32
MDM2 Q00987 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20187636 0.84 HSD17B10 (0.42) ALDH1A1MEN1KMT2APOLBMVD
SCHEMBL22403271 0.81 ALDH1A1 (0.32) ALDH1A1MEN1KMT2APOLBKDM4E
SCHEMBL20200024 0.81 KDM4E (0.43) ALDH1A1MEN1KMT2APOLBSIGMAR1
SCHEMBL20199840 0.80 TACR1 (0.32) ALDH1A1MEN1KMT2APOLBTACR1
SCHEMBL20200035 0.79
SCHEMBL20187501 0.79 ALDH1A1 (0.38) ALDH1A1MEN1KMT2APOLBMVD
SCHEMBL5434193 0.79 HSD17B10 (0.47) ALDH1A1KDM4ETACR1TSHR
SCHEMBL14470272 0.79 HSD17B10 (0.47) ALDH1A1KDM4ETACR1TSHR
SCHEMBL13569369 0.79 HSD17B10 (0.47) ALDH1A1KDM4ETACR1TSHR
SCHEMBL70778 0.78 TSHR (0.46) ALDH1A1KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3544964-B1 HIGH RELAXIVITY GADOLINIUM CHELATE COMPOUNDS FOR USE IN MAGNETIC RESONANCE IMAGING Bayer Pharma AG (DE) 2020-06-17 EP disclosed
WO-2018096082-A1 HIGH RELAXIVITY GADOLINIUM CHELATE COMPOUNDS FOR USE IN MAGNETIC RESONANCE IMAGING BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-31 WO disclosed