SCHEMBL20201431

SCHEMBL20201431

CN1CCC[C@H](P(=O)(O)O)C1=O

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ENO1 P06733 4/20 0.65
BRD4 O60885 1/20 0.34
BRD2 P25440 1/20 0.34
GRM5 P41594 4/20 0.31
DPP4 P27487 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20201424 1.00 ENO1 (0.65) ENO1BRD4BRD2GRM5DPP4
SCHEMBL20201429 0.94 ENO1 (0.58) ENO1BRD4BRD2GRM5DPP4
SCHEMBL20201417 0.94 ENO1 (0.58) ENO1BRD4BRD2GRM5DPP4
SCHEMBL20201428 0.88 ENO1 (0.62) ENO1DPP4
SCHEMBL20201419 0.88 ENO1 (0.62) ENO1DPP4
SCHEMBL18077425 0.78 ENO1 (1.00) ENO1DPP4
SCHEMBL18077428 0.73 ENO1 (0.89) ENO1DPP4
SCHEMBL18077430 0.73 ENO1 (0.89) ENO1DPP4
SCHEMBL25544199 0.72 PIK3CA (0.36) ENO1GRM5
SCHEMBL10598894 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180147219-A1 ENOLASE INHIBITORS AND METHODS OF TREATMENT THEREWITH BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2018-05-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180147219-A1 ENOLASE INHIBITORS AND METHODS OF TREATMENT THEREWITH ENO1, ECE1, ECI1 ENO1 1/4885BRD4 2587/4885BRD2 4224/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.