SCHEMBL20203239

SCHEMBL20203239

Cn1cnc2ncn(CC(=N)OC(=O)NCCc3ccc4ccc(C#N)cc4c3)c(=O)c21

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 14/20 0.54
CDK1 P06493 2/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CCNC P24863 3/20 0.34
CDK8 P49336 3/20 0.34
MAP4K2 Q12851 2/20 0.33
HASPIN Q8TF76 2/20 0.33
CDK19 Q9BWU1 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20203300 0.81 TRPA1 (0.48) TRPA1
SCHEMBL23718270 0.80 TRPA1 (0.52) TRPA1CYP1A2CYP3A4
SCHEMBL20203299 0.80 TRPA1 (0.49) TRPA1
SCHEMBL20203383 0.79 TRPA1 (0.50) TRPA1
SCHEMBL20203409 0.74 TRPA1 (0.52) TRPA1
SCHEMBL29434767 0.70 TRPA1 (1.00) TRPA1
SCHEMBL20187497 0.70 TRPA1 (1.00) TRPA1
SCHEMBL20203276 0.68 TRPA1 (0.41) TRPA1
SCHEMBL22210245 0.66 TRPA1 (0.38) TRPA1
SCHEMBL23718276 0.66 TRPA1 (0.50) TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018096159-A1 OXADIAZOLONES AS TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2018-05-31 WO disclosed