SCHEMBL20209080

SCHEMBL20209080

C=C(c1nc2cc[nH]c2nc1N)n1ccnc1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.37
CD38 P28907 13/20 0.35
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
MAPK1 P28482 2/20 0.31
ADRB2 P07550 2/20 0.30
ADRB1 P08588 2/20 0.30
ADRB3 P13945 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20209088 0.85 CD38 (0.40) CD38
SCHEMBL29625002 0.85 CD38 (0.40) CD38
SCHEMBL20209150 0.74 MAPK1 (0.40) MAPK1
SCHEMBL20935100 0.72 CYP19A1 (0.39) CYP19A1CYP11B1CYP11B2ADRB2ADRB1
SCHEMBL20209076 0.71 MAPK1 (0.37) MAPK1
SCHEMBL20935311 0.69 CYP19A1 (0.38) CYP19A1CYP11B1CYP11B2ADRB2ADRB1
SCHEMBL20208921 0.68 ALDH1A1 (0.41) MAPK1
SCHEMBL23111910 0.67 MAPT (0.41) CD38
SCHEMBL25934515 0.66 MAPK1 (0.50) MAPK1
SCHEMBL20187673 0.66 NPSR1 (0.42) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018096325-A1 BENZODIAZOLIUM COMPOUNDS AS ENAC INHIBITORS Enterprise Therapeutics Limited (GB) 2018-05-31 WO disclosed