SCHEMBL20209435

SCHEMBL20209435

COC(=O)c1ccnc(N[C@@H](C)c2ccccc2)n1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 9/20 0.53
IDH1 O75874 2/20 0.52
CAMK2D Q13557 1/20 0.50
HTR7 P34969 1/20 0.49
HDAC3 O15379 3/20 0.48
HDAC1 Q13547 3/20 0.48
HDAC2 Q92769 3/20 0.48
HDAC6 Q9UBN7 3/20 0.48
LCK P06239 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ASPH Q12797 1/20 0.47
KDM8 Q8N371 1/20 0.47
PLK1 P53350 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30123472 0.87 MAPK14 (0.56) MAPK14IDH1HTR7HDAC3HDAC1
SCHEMBL20187393 0.87 MAPK14 (0.56) MAPK14IDH1HTR7HDAC3HDAC1
SCHEMBL6082153 0.85 MAPK14 (0.54) MAPK14IDH1HTR7HDAC3HDAC1
SCHEMBL6081327 0.80 MAPK14 (0.52) MAPK14HTR7HDAC3HDAC1HDAC2
SCHEMBL6082367 0.78 MAPK14 (0.50) MAPK14HTR7HDAC3HDAC1HDAC2
SCHEMBL6081490 0.78 MAPK14 (0.50) MAPK14HTR7HDAC3HDAC1HDAC2
SCHEMBL670174 0.77 AURKA (0.53) CAMK2D
SCHEMBL6081738 0.77 MAPK14 (0.49) MAPK14HTR7HDAC3HDAC1HDAC2
SCHEMBL20209335 0.76 ADORA2A (0.53) IDH1
SCHEMBL28606159 0.76 ALDH1A1 (0.51) IDH1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110023298-B Isocitrate Dehydrogenase (IDH) inhibitors 浙江迈同生物医药有限公司 2022-12-16 CN disclosed
WO-2018095344-A1 ISOCITRATE DEHYDROGENASE (IDH) INHIBITOR SHANGHAI METON PHARMACEUTICAL CO., LTD (CN) 2018-05-31 WO disclosed