SCHEMBL20187393

SCHEMBL20187393

C[C@H](Nc1nccc(C(=O)O)n1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 8/20 0.56
KDM4E B2RXH2 3/20 0.54
KDM5A P29375 1/20 0.54
JMJD1C Q15652 1/20 0.54
KDM3A Q9Y4C1 1/20 0.54
ASPH Q12797 2/20 0.53
KDM8 Q8N371 2/20 0.53
RIOX2 Q8IUF8 1/20 0.52
HTR7 P34969 1/20 0.52
LDHA P00338 1/20 0.52
LDHB P07195 1/20 0.52
HDAC3 O15379 3/20 0.51
HDAC1 Q13547 3/20 0.51
HDAC2 Q92769 3/20 0.51
HDAC6 Q9UBN7 3/20 0.51
LCK P06239 2/20 0.50
PLK1 P53350 1/20 0.49
IDH1 O75874 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30123472 1.00 MAPK14 (0.56) MAPK14KDM4EKDM5AJMJD1CKDM3A
SCHEMBL6082153 0.89 MAPK14 (0.54) MAPK14HTR7HDAC3HDAC1HDAC2
SCHEMBL20209435 0.87 MAPK14 (0.53) MAPK14KDM4EASPHKDM8HTR7
SCHEMBL6081327 0.83 MAPK14 (0.52) MAPK14HTR7HDAC3HDAC1HDAC2
SCHEMBL6082367 0.81 MAPK14 (0.50) MAPK14HTR7HDAC3HDAC1HDAC2
SCHEMBL6081490 0.81 MAPK14 (0.50) MAPK14HTR7HDAC3HDAC1HDAC2
SCHEMBL6081738 0.80 MAPK14 (0.49) MAPK14HTR7HDAC3HDAC1HDAC2
SCHEMBL6081874 0.78 MAPK14 (0.47) MAPK14KDM4EASPHKDM8HTR7
SCHEMBL14629467 0.78 HTR7 (0.57) MAPK14HTR7LCKPLK1IDH1
SCHEMBL7664862 0.78 LCK (0.54) LCKIDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018095344-A1 ISOCITRATE DEHYDROGENASE (IDH) INHIBITOR SHANGHAI METON PHARMACEUTICAL CO., LTD (CN) 2018-05-31 WO disclosed
WO-2018095344-A1 ISOCITRATE DEHYDROGENASE (IDH) INHIBITOR SHANGHAI METON PHARMACEUTICAL CO., LTD (CN) 2018-05-31 WO disclosed