SCHEMBL20215228

SCHEMBL20215228

O=c1ccn(Cc2ccccc2F)c(-c2cccc(C(F)(F)F)c2Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 12/20 0.42
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.39
NR1H2 P55055 2/20 0.39
NR1H3 Q13133 2/20 0.39
NOTUM Q6P988 1/20 0.36
CHRM5 P08912 1/20 0.35
DPP4 P27487 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
NR1I2 O75469 1/20 0.35
NR3C1 P04150 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20215269 0.92 P2RX7 (0.40) P2RX7NOTUMCHRM5
SCHEMBL20215235 0.92 P2RX7 (0.47) P2RX7NOTUMCHRM5DPP4DPP8
SCHEMBL20215263 0.90 P2RX7 (0.46) P2RX7MAPTTHRBNR1H2NR1H3
SCHEMBL20215255 0.89 GNRHR (0.39) P2RX7NOTUMCHRM5
SCHEMBL20215214 0.88 P2RX7 (0.50) P2RX7MAPT
SCHEMBL20215243 0.88 P2RX7 (0.42) P2RX7NOTUMDPP4DPP8
SCHEMBL20215219 0.86 P2RX7 (0.41) P2RX7MAPTNOTUMDPP4DPP8
SCHEMBL20215275 0.85 P2RX7 (0.44) P2RX7
SCHEMBL20215236 0.85 P2RX7 (0.40) P2RX7
SCHEMBL20215224 0.85 P2RX7 (0.40) P2RX7MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9988373-B2 Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. (JP) 2018-06-05 US disclosed
US-9988373-B2 Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. (JP) 2018-06-05 US disclosed