SCHEMBL20215219

SCHEMBL20215219

O=c1ccn(Cc2ccccc2)c(-c2cccc(C(F)(F)F)c2Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 9/20 0.41
RXFP1 Q9HBX9 2/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 2/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
NOTUM Q6P988 1/20 0.38
DPP4 P27487 1/20 0.38
DPP8 Q6V1X1 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.37
MAPK14 Q16539 2/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20215265 0.93 ALDH1A1 (0.40) P2RX7RXFP1POLBMAPTLMNA
SCHEMBL20215246 0.93 PPARG (0.37) P2RX7RXFP1POLBNOTUMALDH1A1
SCHEMBL20215256 0.92 KDM4E (0.43) P2RX7POLBMAPTLMNATP53
SCHEMBL20215244 0.92 MAPT (0.39) P2RX7POLBMAPTLMNATP53
SCHEMBL20215230 0.91 MAPK14 (0.43) P2RX7POLBMAPTNOTUMMAPK14
SCHEMBL20215253 0.91 MAPT (0.49) P2RX7RXFP1MAPTLMNATP53
SCHEMBL20215239 0.91 P2RX7 (0.38) P2RX7RXFP1MAPTLMNATP53
SCHEMBL20215257 0.91 CHRM5 (0.46) P2RX7MAPTNOTUMDPP8ALDH1A1
SCHEMBL20215217 0.91 P2RX7 (0.43) P2RX7MAPTLMNANOTUMALDH1A1
SCHEMBL20215274 0.90 CHRM5 (0.40) P2RX7RXFP1POLBMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9988373-B2 Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. (JP) 2018-06-05 US disclosed
US-9988373-B2 Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. (JP) 2018-06-05 US disclosed