SCHEMBL20217286

SCHEMBL20217286

COc1ccccc1C(NC(=O)c1ccc(N)c(C(=N)c2ccc(OC3CCN(C)CC3)cc2)c1)C1CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.41
TTK P33981 4/20 0.41
HRH1 P35367 1/20 0.40
CCR3 P51677 1/20 0.40
KCNH2 Q12809 1/20 0.40
AURKB Q96GD4 2/20 0.39
INCENP Q9NQS7 2/20 0.39
F10 P00742 3/20 0.39
KDR P35968 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
ALDH1A1 P00352 2/20 0.37
ACACB O00763 2/20 0.37
SLC5A7 Q9GZV3 3/20 0.36
KMT2A Q03164 2/20 0.36
F2 P00734 1/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
F7 P08709 1/20 0.36
F3 P13726 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20217573 0.91 CYP3A4 (0.41) CYP3A4TTKKCNH2AURKBINCENP
SCHEMBL20217391 0.91 F10 (0.44) CYP3A4TTKHRH1CCR3KCNH2
SCHEMBL20217252 0.91 CYP3A4 (0.41) CYP3A4TTKAURKBINCENPF10
SCHEMBL20217221 0.89 TTK (0.51) CYP3A4TTKAURKBINCENPF10
SCHEMBL20217594 0.88 F10 (0.43) CYP3A4TTKHRH1CCR3KCNH2
SCHEMBL20217751 0.85 CYP3A4 (0.55) CYP3A4TTKAURKBINCENPF10
SCHEMBL20217290 0.85 ALDH1A1 (0.49) CYP3A4TTKAURKBINCENPF10
SCHEMBL20217747 0.83 CYP3A4 (0.47) CYP3A4TTKAURKBINCENPF10
SCHEMBL20217537 0.83 KMT2A (0.43) CYP3A4TTKAURKBINCENPF10
SCHEMBL20217315 0.82 CYP3A4 (0.52) CYP3A4TTKAURKBINCENPF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2766352-B1 INDAZOLE COMPOUNDS AS KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIV HEALTH NETWORK UHN (CA) 2018-06-06 EP disclosed