SCHEMBL20217641

SCHEMBL20217641

N=C(c1ccc(N2CC(N3CCOCC3)C2)cc1)c1cc(C(=O)NC(c2ccccn2)C2CC2)ccc1N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.47
TTK P33981 6/20 0.47
AURKB Q96GD4 6/20 0.47
INCENP Q9NQS7 6/20 0.47
WDR5 P61964 1/20 0.38
SLC6A9 P48067 4/20 0.36
HDAC6 Q9UBN7 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
F10 P00742 2/20 0.34
SCN9A Q15858 1/20 0.33
WDR91 A4D1P6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20217446 0.87 CYP3A4 (0.53) CYP3A4TTKAURKBINCENPWDR5
SCHEMBL20217579 0.84 CYP3A4 (0.65) CYP3A4TTKAURKBINCENPWDR5
SCHEMBL20217371 0.82 CYP3A4 (0.42) CYP3A4TTKAURKBINCENPWDR5
SCHEMBL20217484 0.81 CYP3A4 (0.65) CYP3A4TTKAURKBINCENPSLC6A9
SCHEMBL20217348 0.81 CYP3A4 (0.47) CYP3A4TTKAURKBINCENPSLC6A9
SCHEMBL20217777 0.81 KMT2A (0.49) CYP3A4MAPK1
SCHEMBL20217912 0.81 CYP3A4 (0.43) CYP3A4TTKAURKBINCENPWDR5
SCHEMBL16292275 0.80 TTK (0.73) CYP3A4TTKAURKBINCENP
SCHEMBL14873458 0.80 TTK (0.73) CYP3A4TTKAURKBINCENP
SCHEMBL20217236 0.80 HDAC3 (0.44) HDAC6HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2766352-B1 INDAZOLE COMPOUNDS AS KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIV HEALTH NETWORK UHN (CA) 2018-06-06 EP disclosed