SCHEMBL20217484

SCHEMBL20217484

N=C(c1ccc(N2C3CCC2COC3)cc1)c1cc(C(=O)NC(c2ccccn2)C2CCCC2)ccc1N

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.65
TTK P33981 7/20 0.65
AURKB Q96GD4 7/20 0.65
INCENP Q9NQS7 7/20 0.65
TRPM8 Q7Z2W7 1/20 0.35
SLC6A9 P48067 4/20 0.34
HDAC6 Q9UBN7 1/20 0.34
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 1/20 0.33
CTSS P25774 4/20 0.32
S1PR2 O95136 1/20 0.32
S1PR4 O95977 1/20 0.32
S1PR3 Q99500 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20217579 0.97 CYP3A4 (0.65) CYP3A4TTKAURKBINCENPSLC6A9
SCHEMBL20217446 0.89 CYP3A4 (0.53) CYP3A4TTKAURKBINCENPTRPM8
SCHEMBL20217846 0.86 CYP3A4 (0.49) CYP3A4TTKAURKBINCENPTRPM8
SCHEMBL20217549 0.85 CYP3A4 (0.49) CYP3A4TTKAURKBINCENPMEN1
SCHEMBL20217496 0.82 CYP3A4 (0.62) CYP3A4TTKAURKBINCENPHDAC6
SCHEMBL20217662 0.82 CYP3A4 (0.47) CYP3A4TTKAURKBINCENPTRPM8
SCHEMBL20217641 0.81 CYP3A4 (0.47) CYP3A4TTKAURKBINCENPSLC6A9
SCHEMBL20217348 0.81 CYP3A4 (0.47) CYP3A4TTKAURKBINCENPSLC6A9
SCHEMBL20217458 0.81 CYP3A4 (0.50) CYP3A4TTKAURKBINCENPTRPM8
SCHEMBL20217912 0.81 CYP3A4 (0.43) CYP3A4TTKAURKBINCENPSLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2766352-B1 INDAZOLE COMPOUNDS AS KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIV HEALTH NETWORK UHN (CA) 2018-06-06 EP disclosed