SCHEMBL20217348

SCHEMBL20217348

N=C(c1ccc(CC2CCN(C3COC3)CC2)cc1)c1cc(C(=O)NC(c2ccccn2)C2CC2)ccc1N

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.47
TTK P33981 5/20 0.47
AURKB Q96GD4 5/20 0.47
INCENP Q9NQS7 5/20 0.47
CHRM2 P08172 11/20 0.45
F2 P00734 1/20 0.40
F10 P00742 1/20 0.40
PRSS1 P07477 1/20 0.40
SLC6A9 P48067 1/20 0.35
MCHR1 Q99705 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20217284 0.89 CHRM2 (0.47) CHRM2F2F10PRSS1MCHR1
SCHEMBL20217446 0.85 CYP3A4 (0.53) CYP3A4TTKAURKBINCENPF2
SCHEMBL20217579 0.84 CYP3A4 (0.65) CYP3A4TTKAURKBINCENPSLC6A9
SCHEMBL20217641 0.81 CYP3A4 (0.47) CYP3A4TTKAURKBINCENPF2
SCHEMBL20217484 0.81 CYP3A4 (0.65) CYP3A4TTKAURKBINCENPSLC6A9
SCHEMBL20217912 0.79 CYP3A4 (0.43) CYP3A4TTKAURKBINCENPSLC6A9
SCHEMBL20217549 0.77 CYP3A4 (0.49) CYP3A4TTKAURKBINCENP
SCHEMBL20217478 0.76 LMNA (0.42) CYP3A4TTKAURKBINCENPCHRM2
SCHEMBL20217312 0.76 CYP3A4 (0.40) CYP3A4TTKAURKBINCENPCHRM2
SCHEMBL20217734 0.75 CYP3A4 (0.43) CYP3A4TTKAURKBINCENPCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2766352-B1 INDAZOLE COMPOUNDS AS KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIV HEALTH NETWORK UHN (CA) 2018-06-06 EP disclosed