SCHEMBL20224877

SCHEMBL20224877

Cc1cccn(CCN2CCC(C)(Oc3ccc(Cl)cc3)CC2)c1=O

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 14/20 0.66
L3MBTL1 Q9Y468 1/20 0.38
PKM P14618 1/20 0.36
EPHX2 P34913 1/20 0.36
HTR1A P08908 1/20 0.36
HTR2A P28223 1/20 0.36
HTR7 P34969 1/20 0.36
HTR6 P50406 1/20 0.36
MMP2 P08253 1/20 0.35
MMP3 P08254 1/20 0.35
MMP8 P22894 1/20 0.35
MMP14 P50281 1/20 0.35
MMP17 Q9ULZ9 1/20 0.35
VEGFA P15692 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25462892 0.91 DRD2 (0.56) DRD2EPHX2HTR1AMMP2MMP3
SCHEMBL17848656 0.86 DRD2 (0.63) DRD2
SCHEMBL17848751 0.80 DRD2 (1.00) DRD2L3MBTL1EPHX2HTR1AHTR2A
SCHEMBL17861619 0.77 DRD2 (0.69) DRD2L3MBTL1EPHX2
SCHEMBL17848659 0.76 DRD2 (0.71) DRD2L3MBTL1
SCHEMBL17848638 0.76 DRD2 (0.62) DRD2HTR1A
SCHEMBL17848654 0.75 DRD2 (0.66) DRD2EPHX2HTR1AHTR2AHTR7
SCHEMBL17861621 0.75 DRD2 (0.66) DRD2EPHX2
SCHEMBL17848631 0.74 DRD2 (0.90) DRD2L3MBTL1
SCHEMBL12264162 0.73 DRD2 (0.45) DRD2PKMHTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230143552-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2023-05-11 US disclosed
US-10633336-B2 Dopamine D2 receptor ligands THE BROAD INSTITUTE, INC. (US) 2020-04-28 US disclosed
US-20180155283-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2018-06-07 US disclosed
US-20180155283-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2018-06-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180155283-A1 DOPAMINE D2 RECEPTOR LIGANDS DRD2, DRD3, ARRB1 DRD2 1/4885L3MBTL1 1874/4885PKM 2846/4885
US-10633336-B2 Dopamine D2 receptor ligands DRD2, ARRB1, DRD3 DRD2 1/4885L3MBTL1 2124/4885PKM 3470/4885
US-20230143552-A1 DOPAMINE D2 RECEPTOR LIGANDS DRD2, SLC6A3, NTSR2 DRD2 1/4885L3MBTL1 1719/4885PKM 3719/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.